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Substrates

 

Substrates of CDK5
Substrates Accession No Sites Reference
Amphiphysin 1 NP_001626 Ser272, Ser276, Ser285 Floyd et al., 2001 JBC 276:8104-8110
beta APP P05067 Ser743 Iijima et al., 2000 J. Neurochem. 75:1085-1091
beta catenin A38973   Kesavapany et al., 2001 Eur. J. Neurosci. 13:241-247
Cables AAL83906   Zuckerberg et al., 2000 Neuron 26:633-646
DARPP32 Q9UD71 Thr75 Bibb et al., 1999 Nature 402:669-671
Dab1 = Disabled O75553 Ser491 Keshvara et al., 2002 J. Neuroscience 22:4869-4877
Dynamin 1 NP_004399 Thr480 Tomizawak et al., 2003 JCB 163:813-824
ErbB ??     Fu et al., 2001 Nature Neurosci. 4:374-381
FAK focal adhesion kinase NP_722560 Ser732 Xie et al., 2003 Cell 114:469-482
MAP1B

NP_005900

potential sites:
T667, S2289, S2256
Pigino et al., 1997 J. Cell Sci. 110:257-270
MEF2 A, B, C, D Q14814 (MEF2D) Ser444 Gong et al., 2003 Neuron 38:33-46
MAP2K1, MEK1, MKK1 NP_002746 Thr286 Sharma et al., 2002 JBC 277:528-34
MUNC18 = STXBP1 NP_003156 Thr574 Fletcher et al., 1999 JBC 274:4027-4035
Nestin rat (but not human) NP_006608 Thr 316, Thr 1495 Sahlgreen et al., 2003 MCB 23:5090-5106
Nudel AAF97497   Nisthammer et al., 2000 Neuron 28:697-711
Neurofilament heavy NFH NP_066554 many Lew et al., 1994 Nature 371 423-425
Neurofilament medium NFM NP_005373 many Lew et al., 1994 Nature 371 423-425
NMDA receptors     Wang et al., 2003 Nat Neurosci. 6:1039-1047
p35 (CDK5-activator) NP_003876 Ser8, Thr138, Ser170, Thr197 Patrick et al., 1998 JBC 273:24057-24064
p39 (CDK5-activator) NP_003927 Ser8, Ser173 Humbert et al., 2000 J. Cell Sci. 113:975-983
p53 tumor supressor NP_000537 potentially Ser33, Ser315 Zhang et al., 2002 J. Neurochem. 81:307-313
PAK1 Q13153 Thr212 Nikolic et al., 1998 Nature 395:194-198
Pctaire kinase   Ser95 Cheng et al., 2002 JBC 277:31988-31993
pgamma (PDE regulator) NP_006196 Thr18

Hayashi et al., 2000 JBC 275:32958-32965
Matsuura et al., 2000 JBC 275:32950-32957

PP1-inhibitor Q13522 Ser6, Ser67 Bibb et al., 2001 JBC 276 14490-14497
pRb Retinoblastoma NP_000312 many Lee et al., 1997 JBC 272:5622-5626
Src-tyrosine kinase NP_005408 Ser75 Kato and Maeda 1999 J. Biochem 126:957-961
Synapsin1 NP_008881 Ser553 Matsubara et al., 1996 JBC 271:21108:21113
Tau NP_058519   Baumann et al., 1993 FEBS letters 336:417-424

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axel.knebel@kinasource.co.uk